Asymmetric Total Synthesis of Neooxazolomycin
نویسندگان
چکیده
منابع مشابه
Asymmetric total synthesis of (+)-swainsonine.
A concise asymmetric synthesis of (+)-swainsonine (ent-1) is described starting from 2, which was readily prepared from commercially available l-glutamic acid. The method features installation of the indolizidine ring via an intramolecular cyclisation of α-sulfinyl carbanion as a key step. (+)-Swainsonine was obtained in 11.8% overall yield in 10 steps.
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ژورنال
عنوان ژورنال: Journal of Synthetic Organic Chemistry, Japan
سال: 2020
ISSN: 0037-9980,1883-6526
DOI: 10.5059/yukigoseikyokaishi.78.634